10 and 11) Arylpiperazine derivative of hydantoin with free hydroxyl group 4 or 7 (1.4e3.1 mmol) was slowly refluxed with acetic anhydride (4e10 ml) for 1e20 min. The solution was stored at low temperature for 2e10 days to give a white precipitate of basic form of the product, which was converted into hydrochloride form (10 or 11) by dissolving in methanol and saturation with gaseous HCl ,
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