One-pot preparation of 2-(alkyl)arylbenzoselenazoles from the corresponding N-(acetyl)benzoyl-2-iodoanilines via a microwave-assisted methodology

Sébastien Redon (1) , Youssef Kabri (1) , Maxime D. Crozet (1) , Patrice Vanelle (1)

1 ICR - Institut de Chimie Radicalaire

We report here the first example of a one-pot synthesis of 2-(alkyl)arylbenzoselenazoles from N-(acetyl)benzoyl-2-iodoanilines. The reaction was carried out in the presence of Woollins' reagent under microwave irradiation and resulted in moderate to good yields.

Domains: Chemical Sciences; Organic chemistry

Sébastien Redon, Youssef Kabri, Maxime D. Crozet, Patrice Vanelle. One-pot preparation of 2-(alkyl)arylbenzoselenazoles from the corresponding N-(acetyl)benzoyl-2-iodoanilines via a microwave-assisted methodology. Tetrahedron Letters, 2014, 55 (36), pp.5052-5054. ⟨10.1016/j.tetlet.2014.07.055⟩. ⟨hal-01373020v2⟩